Basic Information
ID: ALA2166531
Type: Functional
Description: Antagonist activity at human H3R-Galphai2-Gbeta1gamma2-RGS4 expressed in Sf9 cells assessed as inhibition of of histamine-induced GTP hydrolysis by steady state GTPase activity assay
Organism: Homo sapiens
Cell type: Sf9
Activity Charts
Bioactivity
Activity Types for Assay ALA2166531
pKb
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 564.79 | 2.15 | 2.15 |
| 592.84 | 2.93 | 2.93 |
| 677.00 | 5.27 | 5.27 |
| 536.73 | 1.53 | 1.53 |
| 564.79 | 2.31 | 2.31 |
| 578.81 | 2.62 | 2.62 |
| 536.73 | 1.37 | 1.37 |