Basic Information
ID: ALA2187699
Type: Binding
Description: Competitive inhibition of human recombinant PACE4 expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate at pH 6.5 after 60 mins by spectrofluorometric analysis
Organism: Homo sapiens
Cell type: S2
Activity Charts
Bioactivity
Activity Types for Assay ALA2187699
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 825.07 | -2.20 | -2.20 |
| 906.06 | -4.56 | -4.56 |
| 983.24 | -4.81 | -4.81 |
| 915.16 | -4.74 | -4.74 |
| 912.16 | -3.66 | -3.66 |
| 941.20 | -4.33 | -4.33 |
| 598.75 | -3.26 | -3.26 |
| 711.91 | -2.73 | -2.73 |
| 938.23 | -1.66 | -1.66 |
| 1051.39 | ||
| 1164.55 | ||
| 1277.71 | ||
| 1051.39 | ||
| 1403.82 | ||
| 1163.61 | ||
| 915.12 | -6.24 | -6.24 |
| 932.05 | -6.19 | -6.19 |