Basic Information
ID: ALA2329083
Type: Binding
Description: Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counting analysis in presence of [gamma-33P]-ATP
Organism: Rattus norvegicus
Activity Charts
Bioactivity
Activity Types for Assay ALA2329083
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 356.18 | 5.18 | 5.18 |
| 355.19 | 3.96 | 3.96 |
| 370.21 | 5.19 | 5.19 |
| 356.18 | 3.42 | 3.42 |
| 400.19 | 3.11 | 3.11 |
| 385.17 | 3.12 | 3.12 |
| 374.27 | 3.38 | 3.38 |
| 371.19 | 2.91 | 2.91 |
| 384.19 | 3.23 | 3.23 |
| 345.28 | 3.67 | 3.67 |
| 335.32 | 2.44 | 2.44 |
| 321.29 | 2.35 | 2.35 |
| 414.22 | 3.20 | 3.20 |
| 403.32 | 3.46 | 3.46 |
| 370.29 | 3.54 | 3.54 |
| 413.32 | 2.85 | 2.85 |
| 389.29 | 3.37 | 3.37 |
| 428.24 | 3.23 | 3.23 |
| 414.22 | 3.14 | 3.14 |
| 321.29 | 2.35 | 2.35 |
| 414.22 | 3.20 | 3.20 |
| 403.32 | 3.46 | 3.46 |
| 400.19 | 3.11 | 3.11 |
| 389.29 | 3.37 | 3.37 |
| 386.20 | 2.91 | 2.91 |
| 399.20 | 3.22 | 3.22 |
| 320.30 | 2.44 | 2.44 |
| 306.28 | 2.36 | 2.36 |
| 399.20 | 3.21 | 3.21 |
| 388.30 | 3.46 | 3.46 |
| 355.28 | 3.55 | 3.55 |
| 398.30 | 2.86 | 2.86 |
| 413.23 | 3.23 | 3.23 |
| 306.28 | 2.36 | 2.36 |
| 399.20 | 3.21 | 3.21 |
| 388.30 | 3.46 | 3.46 |