Basic Information
ID: ALA2330760
Type: Binding
Description: Desensitization of human alpha4beta2 nACHR expressed in HEK293 cells assessed as inhibition of 86Rb+ efflux preincubated for 10 mins measured after 2 hrs by liquid scintillation counting analysis
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA2330760
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 162.24 | 1.85 | 1.85 |
| 211.27 | 1.80 | 1.80 |
| 260.34 | 1.34 | 1.34 |
| 258.36 | 2.67 | 2.67 |
| 272.39 | 3.06 | 3.06 |
| 242.32 | 1.89 | 1.89 |
| 274.36 | 1.64 | 1.64 |
| 276.35 | 2.62 | 2.62 |
| 292.81 | 2.89 | 2.89 |