Basic Information
ID: ALA2331015
Type: Functional
Description: Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hrs by luciferase reporter gene assay
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA2331015
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 103.12 | -0.19 | -0.19 |
| 213.66 | 1.86 | 1.86 |
| 213.66 | 1.86 | 1.86 |
| 444.59 | ||
| 352.38 | 3.67 | 3.67 |
| 362.42 | 4.34 | 4.34 |
| 346.42 | 4.48 | 4.48 |
| 206.19 | 3.29 | 3.29 |
| 376.44 | 5.00 | 5.00 |
| 326.44 | 4.10 | 4.10 |
| 342.34 | 4.40 | 4.40 |
| 304.34 | 4.38 | 4.38 |
| 302.32 | 4.15 | 4.15 |
| 318.36 | 4.60 | 4.60 |
| 288.72 | 3.88 | 3.88 |
| 258.31 | 3.43 | 3.43 |
| 232.27 | 2.73 | 2.73 |
| 330.35 | 3.95 | 3.95 |