Agonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as accumulation of IP1 incubated for 1 hr at 37 degC followed by 15 mins a...

Basic Information

ID: ALA2342579

Type: Functional

Description: Agonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as accumulation of IP1 incubated for 1 hr at 37 degC followed by 15 mins at RT by TR-FRET assay relative to 5HT

Format: BAO_0000219

Organism: Homo sapiens

Cell type: HEK293

Target:  Serotonin 2c (5-HT2c) receptor(ALA225)

Document:  ALA2331121

Agonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as accumulation of IP1 incubated for 1 hr at 37 degC followed by 15 mins at RT by TR-FRET assay relative to 5HT: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
200.281.871.87
198.660.540.54
304.782.122.12
244.291.941.94
244.291.181.18