Basic Information
ID: ALA2351585
Type: Functional
Description: Antagonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated for 15 mins prior to cimaterol induction measured after 5 hrs
Organism: Homo sapiens
Cell type: CHO-K1
Activity Charts
Bioactivity
Activity Types for Assay ALA2351585
Kd
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 494.47 | 2.32 | 2.32 |
| 339.39 | -0.24 | -0.24 |
| 484.55 | 2.22 | 2.22 |
| 492.02 | 3.83 | 3.83 |
| 457.57 | 3.18 | 3.18 |
| 433.51 | 1.96 | 1.96 |
| 527.59 | 3.32 | 3.32 |
| 473.57 | 2.88 | 2.88 |
| 505.57 | 2.35 | 2.35 |
| 372.43 | 1.71 | 1.71 |