Assay Report Card

Basic Information

ID: ALA2379816

Type: Binding

Description: Antagonist activity at human recombinant P2X3 receptor expressed in Xenopus oocytes assessed as inhibition of ATP-induced ion current at 100 nM incubated for 20 mins prior to ATP-induction by two-electrode voltage clamp assay

Organism: Homo sapiens

Cell type: Oocyte

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
511.381.431.43
357.323.043.04
373.322.922.92
473.441.831.83
489.441.721.72
393.382.592.59
409.382.472.47