Assay Report Card

Basic Information

ID: ALA2395412

Type: Binding

Description: Binding affinity to inactivated state of human NaV1.7 channel assessed as inhibition of current evoked by 6 ms depolarizations to 0 mV from holding potential -70 mV at 3 uM by whole-cell patch clamp assay relative to vehicle-treated control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
571.494.104.10