Basic Information
ID: ALA2400933
Type: Binding
Description: Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition measured after 30 mins by liquid scintillation counting analysis
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA2400933
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 374.66 | 2.77 | 2.77 |
| 355.23 | 1.70 | 1.70 |
| 332.79 | 2.73 | 2.73 |
| 468.39 | 2.43 | 2.43 |
| 150.14 | -0.40 | -0.40 |
| 300.32 | 1.17 | 1.17 |
| 312.33 | 1.60 | 1.60 |
| 300.32 | 1.52 | 1.52 |
| 314.35 | 1.83 | 1.83 |
| 319.80 | 1.77 | 1.77 |
| 333.82 | 1.80 | 1.80 |
| 319.80 | 1.77 | 1.77 |
| 333.82 | 2.08 | 2.08 |
| 319.80 | 1.77 | 1.77 |
| 354.24 | 2.42 | 2.42 |
| 349.82 | 1.78 | 1.78 |
| 333.82 | 1.96 | 1.96 |
| 308.77 | 1.03 | 1.03 |
| 326.83 | 0.04 | 0.04 |
| 340.21 | 2.12 | 2.12 |
| 354.24 | 2.42 | 2.42 |
| 340.21 | 2.12 | 2.12 |
| 354.24 | 2.42 | 2.42 |