Basic Information
ID: ALA2401238
Type: Binding
Description: Antagonist activity at human recombinant GABAAalpha1beta2gamma2L receptor expressed in Xenopus laevis assessed as inhibition of GABA-induced chloride current production at 300 uM after 2 to 5 days by two-electrode voltage-clamp electrophysiological assay relative to control
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA2401238
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 126.16 | -0.48 | -0.48 |
| 140.19 | -0.22 | -0.22 |
| 168.24 | 0.56 | 0.56 |
| 196.29 | 1.34 | 1.34 |
| 216.28 | 1.98 | 1.98 |