ID: ALA2438198
Type: Functional
Description: Antagonist activity at human OX2 receptor expressed in HEK cells assessed as inhibition of orexin A-induced Ca2+ accumulation after 1 hr by Fluo-4-AM staining-based FLIPR assay
Organism: Homo sapiens
Cell type: HEK293
Bioactivity
Activity Types for Assay ALA2438198
Ki
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
386.50 | 3.83 | 3.83 |
444.58 | 3.90 | 3.90 |
445.57 | 3.30 | 3.30 |
431.54 | 3.29 | 3.29 |
430.56 | 3.89 | 3.89 |
404.52 | 3.38 | 3.38 |
404.52 | 3.38 | 3.38 |
433.56 | 3.99 | 3.99 |
417.56 | 3.99 | 3.99 |
405.50 | 3.38 | 3.38 |
403.53 | 3.98 | 3.98 |
389.50 | 3.68 | 3.68 |
375.48 | 3.37 | 3.37 |
375.48 | 3.37 | 3.37 |
425.54 | 4.52 | 4.52 |
425.54 | 4.52 | 4.52 |
414.51 | 4.86 | 4.86 |
403.53 | 4.13 | 4.13 |
425.54 | 4.66 | 4.66 |
425.54 | 4.66 | 4.66 |
414.55 | 4.80 | 4.80 |
386.50 | 4.04 | 4.04 |
386.50 | 4.18 | 4.18 |