Assay Report Card

Basic Information

ID: ALA2439243

Type: Binding

Description: Inhibition of GRK2 in HEK293 cells overexpressing human beta2 adrenergic receptor assessed as effect on isoproterenol-induced cAMP production at 1 uM preincubated for 1 hr prior to isoproterenol-stimulation measured after 15 mins by enzyme immunoassay

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
951.14-3.95-3.95