Assay Report Card

Basic Information

ID: ALA2439245

Type: Binding

Description: Inhibition of GRK2 in HEK293 cells overexpressing human beta2 adrenergic receptor assessed as increase in beta2 adrenergic receptor density at 1 uM after 1 hr by gamma counting analysis in presence of [125I]cyanopindolol

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
951.14-3.95-3.95