Basic Information
ID: ALA2444598
Type: Binding
Description: Antagonist activity at human TRPV3 expressed in CHO cells assessed as inhibition of 2APB-induced 45Ca2+ uptake at 1 uM incubated for 10 mins prior to 2APB-challenge measured after 2 to 5 mins by liquid scintillation counting analysis
Organism: Homo sapiens
Cell type: CHO
Activity Charts
Bioactivity
Activity Types for Assay ALA2444598
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 456.85 | 5.12 | 5.12 |
| 456.85 | 5.12 | 5.12 |
| 501.30 | 5.23 | 5.23 |
| 501.30 | 5.23 | 5.23 |
| 440.39 | 4.61 | 4.61 |
| 440.39 | 4.61 | 4.61 |