Basic Information
ID: ALA2444599
Type: Binding
Description: Antagonist activity at human TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced 45Ca2+ uptake incubated for 10 mins prior to capsaicin-challenge measured after 2 to 5 mins by liquid scintillation counting analysis
Organism: Homo sapiens
Cell type: CHO
Activity Charts
Bioactivity
Activity Types for Assay ALA2444599
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 456.85 | 5.12 | 5.12 |
| 456.85 | 5.12 | 5.12 |
| 501.30 | 5.23 | 5.23 |
| 501.30 | 5.23 | 5.23 |
| 440.39 | 4.61 | 4.61 |
| 440.39 | 4.61 | 4.61 |