Basic Information
ID: ALA2445667
Type: Binding
Description: Inhibition of human TRPM8 (unknown origin) expressed in HEK293 cells assessed as inhibition of WS12-induced Ca2+ elevation by FLIPR assay
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA2445667
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 156.27 | 2.44 | 2.44 |
| 311.30 | 2.87 | 2.87 |
| 289.42 | 4.34 | 4.34 |
| 434.54 | 4.93 | 4.93 |
| 377.49 | 3.87 | 3.87 |
| 377.49 | 3.87 | 3.87 |
| 377.49 | 3.87 | 3.87 |
| 386.92 | 4.65 | 4.65 |
| 386.92 | 4.65 | 4.65 |
| 386.92 | 4.65 | 4.65 |
| 386.92 | 4.65 | 4.65 |
| 386.92 | 4.65 | 4.65 |
| 370.47 | 4.14 | 4.14 |
| 370.47 | 4.14 | 4.14 |
| 366.51 | 4.31 | 4.31 |
| 366.51 | 4.31 | 4.31 |
| 352.48 | 4.00 | 4.00 |
| 322.45 | 4.09 | 4.09 |
| 336.48 | 4.01 | 4.01 |
| 318.46 | 3.45 | 3.45 |
| 352.48 | 4.00 | 4.00 |
| 353.47 | 3.39 | 3.39 |
| 353.47 | 3.39 | 3.39 |
| 353.47 | 3.39 | 3.39 |
| 378.52 | 4.39 | 4.39 |
| 366.51 | 4.39 | 4.39 |
| 380.53 | 4.78 | 4.78 |
| 378.52 | 4.53 | 4.53 |
| 364.49 | 4.14 | 4.14 |
| 322.41 | 2.56 | 2.56 |
| 338.45 | 3.61 | 3.61 |
| 366.51 | 4.39 | 4.39 |
| 296.37 | 2.44 | 2.44 |
| 311.39 | 1.90 | 1.90 |
| 324.42 | 3.09 | 3.09 |
| 296.37 | 2.31 | 2.31 |
| 338.45 | 3.48 | 3.48 |
| 310.40 | 2.70 | 2.70 |
| 338.45 | 3.48 | 3.48 |
| 338.45 | 3.61 | 3.61 |
| 338.45 | 3.61 | 3.61 |
| 394.52 | 4.18 | 4.18 |
| 352.48 | 4.00 | 4.00 |
| 352.48 | 4.00 | 4.00 |
| 352.48 | 4.00 | 4.00 |
| 366.49 | 3.93 | 3.93 |
| 396.51 | 3.94 | 3.94 |