Assay Report Card

Basic Information

ID: ALA3089352

Type: Binding

Description: Inhibition of human CB1 receptor internalization expressed in CHO cells assessed as inhibition of [3H]-Win55212-2 uptake preincubated for 1 hr followed by radioligand addition measured after 1 hr by liquid scintillation counting analysis relative to control

Organism: Homo sapiens

Cell type: CHO

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
295.474.134.13
291.433.683.68
263.382.902.90
263.382.902.90
273.424.344.34
289.423.453.45
289.423.453.45
279.381.871.87