Basic Information
ID: ALA3095124
Type: Binding
Description: Inhibition of GLUT1 in human H1299 cells assessed as inhibition of 2-deoxy-D-[3H]-glucose uptake incubated for 15 mins prior to 2-deoxy-D-[3H]-glucose addition measured after 30 mins by liquid scintillation counting analysis
Organism: Homo sapiens
Cell type: H1299
Activity Charts
Bioactivity
Activity Types for Assay ALA3095124
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 274.27 | 2.32 | 2.32 |
| 243.26 | 2.88 | 2.88 |
| 261.25 | 3.02 | 3.02 |
| 277.71 | 3.62 | 3.62 |
| 309.72 | 4.06 | 4.06 |
| 368.32 | 3.68 | 3.68 |