Basic Information
ID: ALA3096231
Type: Functional
Description: Inverse agonist activity at human CB1 receptor expressed in Sf9 cells assessed as stimulation of [35S]GTPgamma binding incubated for 15 mins prior to [35S]GTPgamma addition measured after 35 mins by scintillation proximity assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: Sf9
Target: Cannabinoid CB1 receptor(ALA218)
Document: ALA3091283
Inverse agonist activity at human CB1 receptor expressed in Sf9 cells assessed as stimulation of [35S]GTPgamma binding incubated for 15 mins prior to [35S]GTPgamma addition measured after 35 mins by scintillation proximity assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3096231
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 465.39 | 2.77 | 2.77 |