Agonist activity at human CB1 receptor expressed in Sf9 cells assessed as stimulation of [35S]GTPgamma binding incubated for 15 mins prior to [35S]GTP...

Basic Information

ID: ALA3096234

Type: Functional

Description: Agonist activity at human CB1 receptor expressed in Sf9 cells assessed as stimulation of [35S]GTPgamma binding incubated for 15 mins prior to [35S]GTPgamma addition measured after 35 mins by scintillation proximity assay

Format: BAO_0000219

Organism: Homo sapiens

Cell type: Sf9

Target:  Cannabinoid CB1 receptor(ALA218)

Document:  ALA3091283

Agonist activity at human CB1 receptor expressed in Sf9 cells assessed as stimulation of [35S]GTPgamma binding incubated for 15 mins prior to [35S]GTPgamma addition measured after 35 mins by scintillation proximity assay: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
458.992.912.91
458.992.912.91
453.982.782.78
446.963.043.04
469.033.783.78
443.003.213.21
457.023.473.47
473.023.223.22
469.393.193.19
477.402.912.91
464.402.342.34
490.442.832.83
485.442.252.25
419.363.543.54
449.393.173.17
449.393.173.17
491.474.024.02
463.413.563.56
463.413.563.56
496.973.923.92
496.973.923.92
407.353.133.13
393.323.123.12
423.352.202.20
451.403.243.24