Assay Report Card

Basic Information

ID: ALA3102575

Type: Binding

Description: Reversible inhibition of human recombinant PTP1B expressed in Escherichia coli TB1 using p-nitrophenylphosphate as substrate assessed as residual activity at 25 times IC50 after 1 hr measured after 400 fold dilution

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
463.495.345.34
564.666.826.82
564.666.826.82
550.646.786.78
459.525.245.24
459.525.245.24
489.555.255.25
489.555.255.25
475.525.215.21
475.525.215.21