Assay Report Card

Basic Information

ID: ALA3106504

Type: Binding

Description: Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx at 10 uM preincubated for 30 mins followed by ATP addition by Fluo-4 AM dye-based fluorescence assay

Organism: Homo sapiens

Cell type: 1321-N1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
252.272.642.64
252.273.033.03
251.292.672.67
320.445.555.55
333.444.294.29
320.445.555.55
327.385.655.65