Basic Information
ID: ALA3117036
Type: Binding
Description: Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP incubated for 20 mins prior to addition of fluorescein-labeled GK measured after 2 to 4 hrs by Alpha Screen assay
Format: BAO_0000357
Organism: Homo sapiens
Target: Hexokinase type IV(ALA3820)
Document: ALA3112561
Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP incubated for 20 mins prior to addition of fluorescein-labeled GK measured after 2 to 4 hrs by Alpha Screen assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3117036
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 533.64 | 3.12 | 3.12 |
| 553.62 | 4.13 | 4.13 |
| 567.68 | 2.13 | 2.13 |
| 581.70 | 2.52 | 2.52 |
| 531.62 | 2.73 | 2.73 |
| 545.65 | 3.26 | 3.26 |
| 561.65 | 2.23 | 2.23 |
| 561.65 | 2.23 | 2.23 |
| 561.65 | 2.23 | 2.23 |
| 561.65 | 2.23 | 2.23 |
| 561.65 | 2.23 | 2.23 |
| 561.65 | 2.23 | 2.23 |
| 474.45 | 3.57 | 3.57 |
| 468.42 | 3.51 | 3.51 |
| 489.46 | 3.15 | 3.15 |
| 489.46 | 3.15 | 3.15 |
| 483.43 | 3.09 | 3.09 |
| 483.43 | 3.09 | 3.09 |
| 483.43 | 3.09 | 3.09 |
| 484.42 | 2.49 | 2.49 |
| 484.42 | 2.49 | 2.49 |
| 485.41 | 1.88 | 1.88 |
| 522.47 | 2.88 | 2.88 |
| 522.47 | 2.88 | 2.88 |
| 522.47 | 2.88 | 2.88 |
| 468.50 | 2.34 | 2.34 |
| 468.50 | 2.34 | 2.34 |
| 536.50 | 3.27 | 3.27 |
| 548.51 | 3.27 | 3.27 |
| 564.55 | 3.91 | 3.91 |