Assay Report Card

Basic Information

ID: ALA3128371

Type: Binding

Description: Inhibition of 20s constitutive proteasome beta 2 subunit trypsin-like activity in rabbit erythrocytes using Boc-LRR-AMC as substrate at 100 uM incubated for 15 mins prior to substrate addition measured after 45 mins by fluorescence assay relative to control

Organism: Oryctolagus cuniculus

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
252.300.650.65
333.183.183.18
286.331.711.71
305.381.151.15
284.383.323.32
307.421.801.80
366.875.025.02
401.325.675.67
178.191.071.07