Basic Information
ID: ALA3128372
Type: Binding
Description: Inhibition of 20s constitutive proteasome beta 2 subunit trypsin-like activity in rabbit erythrocytes using Boc-LRR-AMC as substrate incubated for 15 mins prior to substrate addition measured after 45 mins by fluorescence assay
Organism: Oryctolagus cuniculus
Activity Charts
Bioactivity
Activity Types for Assay ALA3128372
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 313.78 | 1.13 | 1.13 |
| 218.26 | 1.99 | 1.99 |
| 246.31 | 2.48 | 2.48 |
| 288.73 | 3.88 | 3.88 |
| 333.37 | 1.88 | 1.88 |
| 328.37 | 2.34 | 2.34 |
| 342.40 | 2.65 | 2.65 |
| 346.36 | 2.48 | 2.48 |
| 362.81 | 2.99 | 2.99 |
| 247.32 | 2.06 | 2.06 |
| 231.29 | 2.12 | 2.12 |
| 253.30 | 1.26 | 1.26 |
| 257.29 | 1.82 | 1.82 |
| 213.19 | 1.63 | 1.63 |
| 177.16 | 0.79 | 0.79 |
| 178.19 | 0.95 | 0.95 |
| 240.26 | 2.09 | 2.09 |
| 204.23 | 1.49 | 1.49 |
| 232.28 | 1.89 | 1.89 |
| 222.24 | 0.42 | 0.42 |
| 321.38 | 0.12 | 0.12 |
| 328.37 | 1.87 | 1.87 |
| 318.83 | 3.97 | 3.97 |
| 298.41 | 3.63 | 3.63 |
| 366.87 | 5.02 | 5.02 |
| 357.48 | 2.83 | 2.83 |
| 179.17 | 1.19 | 1.19 |
| 219.24 | 2.12 | 2.12 |
| 195.24 | 1.78 | 1.78 |
| 235.31 | 2.70 | 2.70 |
| 177.20 | 1.80 | 1.80 |
| 217.27 | 2.72 | 2.72 |
| 192.22 | 1.46 | 1.46 |