Assay Report Card

Basic Information

ID: ALA3128969

Type: Binding

Description: Reversible inhibition of N-terminal GST-tagged recombinant human Histone-lysine N-methyltransferase G9a using S-(5'-adenosyl)-L-methionine chloride as substrate assessed as enzyme recovery at 10 fold IC50 preincubated for 30 mins followed by 100 fold dilution in presence of DTT

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
696.861.331.33
356.473.103.10