Basic Information
ID: ALA3131528
Type: Binding
Description: Inhibition of biotin-tagged human GKRP-fluorescein-tagged human GK interaction preincubated for 20 mins followed by fluorescein-tagged human GK addition measured after 2 to 4 hrs by AlphaScreen assay
Format: BAO_0000357
Organism: Homo sapiens
Target: Glucokinase regulatory protein(ALA1075152)
Document: ALA3124752
Inhibition of biotin-tagged human GKRP-fluorescein-tagged human GK interaction preincubated for 20 mins followed by fluorescein-tagged human GK addition measured after 2 to 4 hrs by AlphaScreen assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3131528
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 533.64 | 3.12 | 3.12 |
| 474.45 | 3.57 | 3.57 |
| 580.57 | 4.89 | 4.89 |
| 580.57 | 4.89 | 4.89 |
| 578.60 | 5.49 | 5.49 |
| 578.60 | 5.49 | 5.49 |
| 578.60 | 5.49 | 5.49 |
| 565.56 | 4.58 | 4.58 |
| 570.62 | 5.91 | 5.91 |
| 572.59 | 4.76 | 4.76 |
| 573.58 | 3.27 | 3.27 |
| 587.61 | 3.66 | 3.66 |
| 518.62 | 4.21 | 4.21 |
| 518.62 | 4.21 | 4.21 |
| 533.64 | 3.12 | 3.12 |
| 488.48 | 3.96 | 3.96 |
| 488.48 | 3.96 | 3.96 |
| 488.48 | 3.96 | 3.96 |
| 488.48 | 3.96 | 3.96 |
| 502.50 | 4.35 | 4.35 |
| 516.53 | 4.60 | 4.60 |
| 550.55 | 5.31 | 5.31 |
| 564.57 | 5.18 | 5.18 |
| 580.57 | 4.89 | 4.89 |