Basic Information
ID: ALA3225545
Type: Functional
Description: Antagonist activity at human recombinant histamine H2 receptor-Gsalphas fusion protein expressed in Sf9 cells assessed as inhibition of histamine-induced [35S]GTPgammaS binding after 90 mins by liquid scintillation counting
Organism: Homo sapiens
Cell type: Sf9
Activity Charts
Bioactivity
Activity Types for Assay ALA3225545
pKb
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 252.35 | 0.60 | 0.60 |
| 370.49 | 1.67 | 1.67 |
| 234.31 | 0.69 | 0.69 |
| 220.28 | 0.30 | 0.30 |
| 342.47 | 2.46 | 2.46 |
| 234.31 | 0.69 | 0.69 |
| 356.50 | 2.85 | 2.85 |
| 343.46 | 1.94 | 1.94 |
| 356.46 | 1.28 | 1.28 |
| 248.33 | 1.01 | 1.01 |
| 370.53 | 3.17 | 3.17 |
| 236.28 | -0.64 | -0.64 |
| 358.48 | 1.52 | 1.52 |
| 237.27 | -1.17 | -1.17 |
| 359.46 | 1.00 | 1.00 |
| 373.49 | 1.39 | 1.39 |
| 254.32 | -0.48 | -0.48 |
| 376.52 | 1.68 | 1.68 |
| 354.48 | 2.69 | 2.69 |
| 368.51 | 3.08 | 3.08 |
| 356.46 | 1.28 | 1.28 |