Assay Report Card

Basic Information

ID: ALA3225547

Type: Functional

Description: Intrinsic activity at human recombinant histamine H3 receptor expressed in Sf9 cells coexpressing Galphai2,Gbeta1gamma2 and RGS4 assessed as [35S]GTPgammaS binding at 10 uM after 90 mins by liquid scintillation counting relative to histamine

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
342.472.542.54
370.491.671.67
234.310.690.69
356.502.852.85
220.280.300.30
342.472.462.46
234.310.690.69
356.502.852.85
356.461.281.28
248.331.011.01
370.533.173.17
232.290.530.53
354.482.692.69
246.320.920.92
368.513.083.08
234.27-0.88-0.88
356.461.281.28
248.29-0.49-0.49