Basic Information
ID: ALA3225551
Type: Functional
Description: Agonist activity at human recombinant histamine H3 receptor expressed in Sf9 cells coexpressing Galphai2,Gbeta1gamma2 and RGS4 assessed as [35S]GTPgammaS binding after 90 mins by liquid scintillation counting
Organism: Homo sapiens
Cell type: Sf9
Activity Charts
Bioactivity
Activity Types for Assay ALA3225551
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 252.35 | 0.60 | 0.60 |
| 111.15 | -0.09 | -0.09 |
| 234.31 | 0.69 | 0.69 |
| 221.27 | -0.23 | -0.23 |
| 343.46 | 1.94 | 1.94 |
| 236.28 | -0.64 | -0.64 |
| 358.48 | 1.52 | 1.52 |
| 237.27 | -1.17 | -1.17 |
| 359.46 | 1.00 | 1.00 |
| 251.30 | -0.77 | -0.77 |
| 373.49 | 1.39 | 1.39 |
| 254.32 | -0.48 | -0.48 |
| 376.52 | 1.68 | 1.68 |