Assay Report Card

Basic Information

ID: ALA3225557

Type: Binding

Description: Intrinsic activity at human recombinant histamine H3 receptor expressed in Sf9 cells coexpressing Galphai2,Gbeta1gamma2 and RGS4 preincubated for 2 mins before [gamma32P]GTP addition measured after 20 mins by steady-state GTPase activity assay relative to histamine

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
313.401.971.97
375.482.932.93
313.411.971.97
319.432.032.03
375.483.003.00
382.492.452.45
313.411.971.97
375.483.003.00
314.391.361.36
376.462.392.39
323.443.243.24
385.514.274.27
324.432.642.64
386.503.673.67
324.432.642.64
386.503.673.67
324.432.642.64
386.503.673.67
370.502.902.90
376.532.962.96
432.573.933.93
439.593.383.38
313.411.901.90