Basic Information
ID: ALA3225910
Type: Binding
Description: Agonist activity at human recombinant histamine H1 receptor expressed in Sf9 cells coexpressing RGS4 preincubated for 2 mins before [gamma32P]GTP addition measured after 20 mins by steady-state GTPase activity assay
Organism: Homo sapiens
Cell type: Sf9
Activity Charts
Bioactivity
Activity Types for Assay ALA3225910
pEC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 252.35 | 0.60 | 0.60 |
| 111.15 | -0.09 | -0.09 |
| 292.45 | 2.80 | 2.80 |
| 319.43 | 2.03 | 2.03 |
| 382.49 | 2.45 | 2.45 |
| 313.41 | 1.97 | 1.97 |
| 314.39 | 1.36 | 1.36 |
| 220.28 | 0.30 | 0.30 |
| 221.27 | -0.23 | -0.23 |
| 236.28 | -0.64 | -0.64 |
| 237.27 | -1.17 | -1.17 |
| 359.46 | 1.00 | 1.00 |
| 251.30 | -0.77 | -0.77 |
| 373.49 | 1.39 | 1.39 |
| 254.32 | -0.48 | -0.48 |
| 376.52 | 1.68 | 1.68 |
| 232.29 | 0.53 | 0.53 |
| 234.27 | -0.88 | -0.88 |
| 324.43 | 2.64 | 2.64 |
| 376.53 | 2.96 | 2.96 |
| 439.59 | 3.38 | 3.38 |
| 313.41 | 1.90 | 1.90 |