Assay Report Card

Basic Information

ID: ALA3227487

Type: Functional

Description: Antagonist activity at CCR5 in Gqi5 transfected human MOLT4 cells assessed as inhibition of RANTES-stimulated Ca2+ influx preincubated for 15 mins followed by DAMGO challenge

Organism: Homo sapiens

Cell type: MOLT-4

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
513.685.955.95
1197.48
886.104.854.85
528.695.535.53
628.817.307.30
657.814.654.65