Basic Information
ID: ALA3238730
Type: Binding
Description: Antagonist activity at rat TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced Ca2+ influx incubated 2.5 mins prior to icilin challenge by luminometry
Organism: Rattus norvegicus
Cell type: CHO
Activity Charts
Bioactivity
Activity Types for Assay ALA3238730
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 414.40 | 6.02 | 6.02 |
| 414.40 | 6.02 | 6.02 |
| 440.42 | 5.58 | 5.58 |
| 421.42 | 5.76 | 5.76 |
| 421.42 | 5.76 | 5.76 |
| 421.42 | 5.76 | 5.76 |
| 397.40 | 5.28 | 5.28 |
| 397.40 | 5.28 | 5.28 |
| 397.40 | 5.28 | 5.28 |
| 376.42 | 5.16 | 5.16 |
| 362.39 | 4.77 | 4.77 |
| 416.37 | 5.31 | 5.31 |
| 416.37 | 5.31 | 5.31 |
| 478.44 | 6.67 | 6.67 |
| 428.43 | 6.20 | 6.20 |
| 450.38 | 6.57 | 6.57 |
| 415.39 | 5.42 | 5.42 |
| 415.39 | 5.42 | 5.42 |
| 415.39 | 5.42 | 5.42 |
| 415.39 | 5.42 | 5.42 |
| 416.38 | 4.81 | 4.81 |
| 416.38 | 4.81 | 4.81 |
| 398.39 | 4.68 | 4.68 |
| 422.41 | 5.15 | 5.15 |
| 417.35 | 4.71 | 4.71 |
| 417.35 | 4.71 | 4.71 |
| 434.36 | 5.45 | 5.45 |
| 435.34 | 4.85 | 4.85 |