ID: ALA3238809
Type: Binding
Description: Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane potential blue assay
Organism: Mus musculus
Cell type: HEK293
Bioactivity
Activity Types for Assay ALA3238809
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
260.13 | 1.09 | 1.09 |
193.25 | 1.39 | 1.39 |
207.27 | 1.69 | 1.69 |
191.23 | 1.40 | 1.40 |
263.38 | 3.42 | 3.42 |
287.40 | 3.35 | 3.35 |
271.36 | 3.06 | 3.06 |
273.38 | 3.05 | 3.05 |
273.38 | 3.05 | 3.05 |
340.26 | 2.75 | 2.75 |
233.31 | 2.40 | 2.40 |
217.27 | 2.11 | 2.11 |
219.28 | 2.09 | 2.09 |
219.28 | 2.09 | 2.09 |
286.17 | 1.79 | 1.79 |
193.25 | 1.39 | 1.39 |
235.33 | 2.64 | 2.64 |
289.42 | 3.81 | 3.81 |
283.37 | 3.28 | 3.28 |
313.40 | 3.29 | 3.29 |
343.42 | 3.30 | 3.30 |