Assay Report Card

Basic Information

ID: ALA3292904

Type: Binding

Description: Inhibition of CTR in Plasmodium falciparum C4Dd2 expressing chloroquine-resistance-conferring pfcrt alleles assessed as increase of accumulation of [3H]-chloroquine level at 1 uM after 1 hr relative to control

Organism: Plasmodium falciparum

Strain: C4Dd2

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
454.615.095.09
274.803.823.82
300.834.514.51
288.824.214.21
302.854.604.60
206.253.043.04