Basic Information
ID: ALA3299556
Type: Binding
Description: Antagonist activity at human TRPM8 expressed in CHOK1 cells assessed as inhibition of menthol-induced calcium flux incubated 10 mins prior to menthol addition by FLIPR assay relative to control
Organism: Homo sapiens
Cell type: CHO-K1
Activity Charts
Bioactivity
Activity Types for Assay ALA3299556
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 262.23 | 4.25 | 4.25 |
| 296.68 | 4.90 | 4.90 |
| 276.26 | 4.56 | 4.56 |
| 292.26 | 4.26 | 4.26 |
| 332.33 | 5.04 | 5.04 |
| 346.23 | 5.15 | 5.15 |