Assay Report Card

Basic Information

ID: ALA3368171

Type: Binding

Description: Inhibition of HIV-1 protease using DABCYL-Abu-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-EDANS as substrate preincubated at 10 uM for 15 mins before substrate addition measured over 15 mins by fluorometric assay

Organism: Human immunodeficiency virus 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
685.901.471.47
346.380.120.12
527.622.392.39
390.441.501.50
408.502.672.67
465.550.890.89
394.472.282.28
434.543.203.20
422.532.912.91
403.440.440.44
330.381.151.15
362.430.660.66
320.35-0.36-0.36
320.35-0.36-0.36
422.481.611.61
452.552.272.27
470.574.174.17
471.562.592.59
409.491.091.09
420.512.762.76
436.511.731.73
410.471.251.25
366.421.501.50
344.411.591.59
375.43-0.72-0.72
354.400.450.45
354.400.450.45
459.540.870.87
473.570.910.91
400.470.050.05
368.430.680.68
368.430.540.54
368.430.680.68