Basic Information
ID: ALA3376222
Type: Functional
Description: Antagonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP at 100 uM by scintillation counting in presence of 30 nM CP55940 (Rvb = 0 +/- 5%)
Organism: Homo sapiens
Cell type: Sf9
Activity Charts
Bioactivity
Activity Types for Assay ALA3376222
Emax
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 504.37 | 4.13 | 4.13 |
| 476.06 | 6.81 | 6.81 |
| 421.59 | 5.55 | 5.55 |
| 407.56 | 5.31 | 5.31 |
| 380.49 | 4.86 | 4.86 |
| 534.79 | 7.19 | 7.19 |
| 436.60 | 4.46 | 4.46 |
| 1010.47 | ||
| 814.09 | 8.74 | 8.74 |
| 842.14 | 9.52 | 9.52 |
| 548.82 | 7.48 | 7.48 |
| 450.63 | 4.75 | 4.75 |
| 1038.52 | ||
| 842.14 | 9.33 | 9.33 |