Basic Information
ID: ALA3378196
Type: Binding
Description: Inhibition of SETD8 (unknown origin) catalytic domain expressed in Escherichia coli using biotinylated H4 (1-24) peptide substrate after 1 hr by scintillation proximity assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3378196
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 413.57 | 3.93 | 3.93 |
| 371.49 | 2.75 | 2.75 |
| 385.51 | 3.15 | 3.15 |
| 399.54 | 3.54 | 3.54 |
| 427.59 | 4.32 | 4.32 |
| 387.53 | 3.39 | 3.39 |
| 415.58 | 4.17 | 4.17 |
| 528.70 | 4.38 | 4.38 |
| 428.58 | 2.73 | 2.73 |
| 442.61 | 3.08 | 3.08 |
| 456.64 | 3.47 | 3.47 |
| 470.66 | 3.86 | 3.86 |
| 427.55 | 3.45 | 3.45 |
| 427.59 | 3.95 | 3.95 |
| 427.59 | 4.32 | 4.32 |
| 441.62 | 4.71 | 4.71 |
| 387.53 | 3.39 | 3.39 |
| 428.58 | 2.73 | 2.73 |
| 442.61 | 3.08 | 3.08 |
| 441.62 | 4.70 | 4.70 |
| 455.65 | 5.09 | 5.09 |
| 427.59 | 4.68 | 4.68 |
| 441.62 | 5.07 | 5.07 |
| 378.90 | 3.98 | 3.98 |