Basic Information
ID: ALA3384241
Type: Binding
Description: Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition by fluorescence assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3384241
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 174.20 | 1.99 | 1.99 |
| 213.71 | 1.82 | 1.82 |
| 253.77 | 2.75 | 2.75 |
| 279.81 | 2.92 | 2.92 |
| 239.75 | 1.99 | 1.99 |
| 309.84 | 2.93 | 2.93 |
| 269.77 | 2.00 | 2.00 |
| 253.77 | 2.55 | 2.55 |
| 267.80 | 2.61 | 2.61 |
| 245.78 | 2.05 | 2.05 |
| 283.80 | 2.75 | 2.75 |
| 243.73 | 1.83 | 1.83 |
| 283.80 | 2.75 | 2.75 |
| 243.73 | 1.83 | 1.83 |
| 241.76 | 2.46 | 2.46 |
| 225.72 | 1.60 | 1.60 |
| 265.78 | 2.53 | 2.53 |
| 293.72 | 2.62 | 2.62 |
| 239.75 | 1.91 | 1.91 |
| 239.75 | 1.91 | 1.91 |
| 239.75 | 1.99 | 1.99 |
| 260.16 | 2.26 | 2.26 |
| 304.62 | 2.37 | 2.37 |
| 255.75 | 1.61 | 1.61 |
| 255.75 | 1.61 | 1.61 |
| 285.77 | 1.62 | 1.62 |
| 158.20 | 2.29 | 2.29 |
| 158.20 | 2.29 | 2.29 |
| 178.62 | 2.64 | 2.64 |
| 223.07 | 2.74 | 2.74 |
| 174.20 | 1.99 | 1.99 |
| 204.22 | 2.00 | 2.00 |