Basic Information
ID: ALA3387265
Type: Functional
Description: Reversible antagonist activity against human thromboxane A2 receptor alpha expressed in QBI-HEK293A cells assessed as reduction in I-BOP-induced inositol monophosphate production at 1 uM incubated for 15 to 60 mins before I-BOP addition and measured after 6 consecutive drug washout by HTRF assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: HEK293-A
Target: Thromboxane A2 receptor(ALA2069)
Document: ALA3351871
Reversible antagonist activity against human thromboxane A2 receptor alpha expressed in QBI-HEK293A cells assessed as reduction in I-BOP-induced inositol monophosphate production at 1 uM incubated for 15 to 60 mins before I-BOP addition and measured after 6 consecutive drug washout by HTRF assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3387265
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 379.87 | 2.80 | 2.80 |