Assay Report Card

Basic Information

ID: ALA3398874

Type: Binding

Description: Antagonist activity against human recombinant TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced Ca2+ influx pre-treated 5 mins before capsaicin addition by Fluo-4 dye based assay

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
305.423.793.79
318.423.803.80
442.657.097.09
458.656.066.06
576.787.867.86