ID: ALA3398874
Type: Binding
Description: Antagonist activity against human recombinant TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced Ca2+ influx pre-treated 5 mins before capsaicin addition by Fluo-4 dye based assay
Organism: Homo sapiens
Cell type: HEK293
Bioactivity
Activity Types for Assay ALA3398874
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
305.42 | 3.79 | 3.79 |
318.42 | 3.80 | 3.80 |
442.65 | 7.09 | 7.09 |
458.65 | 6.06 | 6.06 |
576.78 | 7.86 | 7.86 |