Assay Report Card

Basic Information

ID: ALA3404114

Type: Binding

Description: Inhibition of human CHT Leu530Ala and Val531Ala mutant expressed in HEK293 cells assessed as remaining transporter activity in presence of 10 uM [3H]choline by [3H]choline uptake assay

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
415.533.993.99
386.502.612.61
428.583.713.71
400.523.093.09
389.542.772.77
290.322.442.44
402.564.254.25
384.482.672.67
400.522.922.92
358.444.064.06
403.553.643.64
403.553.643.64
411.553.703.70
372.474.454.45
387.483.213.21
375.473.073.07
387.483.213.21
401.513.603.60
403.482.452.45
373.452.872.87
387.483.213.21
346.433.773.77