ID: ALA3404114
Type: Binding
Description: Inhibition of human CHT Leu530Ala and Val531Ala mutant expressed in HEK293 cells assessed as remaining transporter activity in presence of 10 uM [3H]choline by [3H]choline uptake assay
Organism: Homo sapiens
Cell type: HEK293
Bioactivity
Activity Types for Assay ALA3404114
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
415.53 | 3.99 | 3.99 |
386.50 | 2.61 | 2.61 |
428.58 | 3.71 | 3.71 |
400.52 | 3.09 | 3.09 |
389.54 | 2.77 | 2.77 |
290.32 | 2.44 | 2.44 |
402.56 | 4.25 | 4.25 |
384.48 | 2.67 | 2.67 |
400.52 | 2.92 | 2.92 |
358.44 | 4.06 | 4.06 |
403.55 | 3.64 | 3.64 |
403.55 | 3.64 | 3.64 |
411.55 | 3.70 | 3.70 |
372.47 | 4.45 | 4.45 |
387.48 | 3.21 | 3.21 |
375.47 | 3.07 | 3.07 |
387.48 | 3.21 | 3.21 |
401.51 | 3.60 | 3.60 |
403.48 | 2.45 | 2.45 |
373.45 | 2.87 | 2.87 |
387.48 | 3.21 | 3.21 |
346.43 | 3.77 | 3.77 |