Basic Information
ID: ALA3417975
Type: Binding
Description: Inhibition of rat brain synaptosomes GAT1 assessed as inhibition of [3H]GABA uptake by liquid scintillation counting
Organism: Rattus norvegicus
Tissue: Brain
Subcellular Fraction: Synaptosomes
Activity Charts
Bioactivity
Activity Types for Assay ALA3417975
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 333.43 | 4.29 | 4.29 |
| 375.56 | 5.04 | 5.04 |
| 367.49 | 4.02 | 4.02 |
| 352.43 | 3.25 | 3.25 |
| 365.52 | 5.18 | 5.18 |
| 391.56 | 4.63 | 4.63 |
| 353.42 | 2.65 | 2.65 |