Assay Report Card

Basic Information

ID: ALA3418218

Type: Binding

Description: Inhibition of human recombinant ERAP1 expressed in baculovirus infected Sf9 cells using L-leucine-7-amido-4-methyl coumarin as substrate up to 100 uM after 5 to 10 mins by fluorescence assay

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
419.483.143.14
405.453.053.05
329.361.271.27
433.513.533.53
279.341.371.37
265.311.281.28
322.37-0.42-0.42
308.34-0.50-0.50
441.531.181.18
427.511.091.09
427.511.091.09
443.500.790.79
471.561.151.15
407.520.980.98
504.592.982.98
414.461.321.32
364.451.561.56
407.48-0.36-0.36
419.483.143.14
329.361.271.27
279.341.371.37
279.341.511.51
322.37-0.42-0.42
329.361.071.07
428.493.423.42
455.561.571.57
502.623.673.67
412.492.012.01
582.663.583.58
695.826.316.31
407.520.980.98
364.451.561.56
407.521.131.13
450.54-0.80-0.80