Basic Information
ID: ALA3418221
Type: Binding
Description: Inhibition of human recombinant ERAP2 expressed in baculovirus infected cabbage looper ovary Hi5 cells using L-arginyl-7-amido-4-methyl coumarin as substrate after 5 to 10 mins by fluorescence assay
Organism: Homo sapiens
Tissue: Female gonad
Cell type: BTI-TN-5B1-4
Activity Charts
Bioactivity
Activity Types for Assay ALA3418221
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 329.36 | 1.27 | 1.27 |
| 315.33 | 1.18 | 1.18 |
| 279.34 | 1.51 | 1.51 |
| 322.37 | -0.42 | -0.42 |
| 308.34 | -0.50 | -0.50 |
| 427.51 | 1.09 | 1.09 |
| 443.50 | 0.79 | 0.79 |
| 471.56 | 1.27 | 1.27 |
| 561.68 | 3.15 | 3.15 |
| 407.52 | 0.98 | 0.98 |
| 393.49 | 0.89 | 0.89 |
| 407.52 | 1.13 | 1.13 |
| 450.54 | -0.80 | -0.80 |
| 504.59 | 2.98 | 2.98 |
| 414.46 | 1.32 | 1.32 |
| 492.53 | 1.70 | 1.70 |
| 430.46 | 0.14 | 0.14 |
| 591.67 | 4.05 | 4.05 |
| 501.54 | 2.39 | 2.39 |
| 695.82 | 6.31 | 6.31 |
| 515.57 | 2.78 | 2.78 |
| 454.57 | 3.22 | 3.22 |
| 364.45 | 1.56 | 1.56 |
| 442.52 | 1.94 | 1.94 |
| 541.65 | 4.29 | 4.29 |
| 451.53 | 2.63 | 2.63 |
| 435.53 | 0.26 | 0.26 |
| 407.48 | -0.36 | -0.36 |
| 485.55 | 0.02 | 0.02 |
| 494.56 | 0.70 | 0.70 |
| 327.38 | 1.95 | 1.95 |
| 329.36 | 1.27 | 1.27 |
| 279.34 | 1.37 | 1.37 |
| 279.34 | 1.51 | 1.51 |
| 322.37 | -0.42 | -0.42 |
| 428.49 | 3.42 | 3.42 |
| 338.37 | 1.76 | 1.76 |
| 502.62 | 3.67 | 3.67 |
| 412.49 | 2.01 | 2.01 |
| 490.56 | 2.39 | 2.39 |
| 589.70 | 4.73 | 4.73 |
| 483.57 | 0.70 | 0.70 |
| 582.66 | 3.58 | 3.58 |
| 492.53 | 1.70 | 1.70 |
| 681.79 | 5.92 | 5.92 |
| 501.54 | 2.39 | 2.39 |
| 457.53 | 0.88 | 0.88 |
| 695.82 | 6.31 | 6.31 |
| 515.57 | 2.78 | 2.78 |
| 541.65 | 4.15 | 4.15 |
| 454.57 | 3.22 | 3.22 |
| 364.45 | 1.56 | 1.56 |
| 442.52 | 1.94 | 1.94 |
| 541.65 | 4.29 | 4.29 |
| 451.53 | 2.63 | 2.63 |
| 407.52 | 1.13 | 1.13 |
| 485.55 | 0.02 | 0.02 |
| 494.56 | 0.70 | 0.70 |
| 450.54 | -0.80 | -0.80 |
| 512.59 | 3.53 | 3.53 |