Assay Report Card

Basic Information

ID: ALA3420660

Type: Binding

Description: Competitive antagonist activity at recombinant human P2X7 receptor expressed in HEK293 cells assessed as inhibition of BzATP-induced intracellular ethidium bromide uptake at 0.1 to 1 uM after 2 hrs by fluorescence assay in presence of BzATP

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
687.105.445.44