Assay Report Card

Basic Information

ID: ALA3532959

Type: ADME

Description: Antagonist activity at human CAR expressed in human HepG2 cells coexpressing CYP2B6 assessed as inhibition of CITCO-induced receptor activation up to 100 uM after 24 hrs by dual luciferase reporter gene assay

Organism: Homo sapiens

Cell type: HepG2

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
326.30-0.74-0.74